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Endomorphin-1
添加购物车| 名称 | Endomorphin-1 |
|---|---|
| CAS No. | 189388-22-5 |
| 目录号 | ONP10633 |
| 规格 | mg/g |
| 纯度 | ≥98% |
| 价格 | 更多在线询价 |
| 贮存 | -20°C |
| 分子量 | 610.7 |
| 序列结构 | H-TYR-PRO-TRP-PHE-OH-NH2 |
| 库存 | |
| 产品简述 | Endomorphin-1 (EM-1) is a recently isolated endogenous peptide having potent analgesic activity and high affinity and selectivity for the mu-opioid receptor. Endomorphin-1 activates G proteins and inhibits adenylyl cyclase activity in membrane preparations from cells stably expressing the mu opioid receptor, an effect reversed by the mu receptor antagonist CTAP (D-Phe-Cys-Tyr-D-Trp-Arg-Thr-Pen-Thr-NH2). However, endomorphin-1 appears to have no influence on cells stably expressing the delta opioid receptor. |