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Men 10376
添加购物车| 名称 | Men 10376 |
|---|---|
| CAS No. | 135306-85-3 |
| 目录号 | ONP10615 |
| 规格 | mg/g |
| 纯度 | ≥98% |
| 价格 | 更多在线询价 |
| 贮存 | -20°C |
| 分子量 | 1081.22 |
| 序列结构 | H-ASP-TYR-d-TRP-VAL-d-TRP-d-TRP-LYS-OH-NH2 |
| 库存 | |
| 产品简述 | Men 10376 is a potent and selective NK2 tachykinin receptor antagonist. MEN 10376 was devoid of significant agonist activity at i.v. doses (1-3 mumol/kg) which selectively antagonized the effects of an NK-2 agonist [beta-Ala8]-neurokinin A(4-10) (bladder contraction in rats, bronchoconstriction in guinea pigs) without affecting the response to an NK-1 agonist [Sar9]-substance P sulfone (hypotension, salivation and bladder contraction in rats, bronchoconstriction in guinea pigs). |